Table 6 KD* values obtained for each of the conjugates upon binding to the NOP receptor
Peptide/Conjugate | KD (μM) |
|---|---|
Pomolate-MiF-1 | 72 ± 3.4 |
Betanin-Tri-MiF-1 | 25.1 ± 4.7 |
Sinapate-MiF-1 | Could not be determined |
Gallate-MiF-1 | 41 ± 2.1 |
MiF-1 | 98.5 ± 3.2 |
Pomolate-NPFF | 39.2 ± 5.3 |
Betanin-Tri-NPFF | 17.3 ± 4.0 |
Sinapate-NPFF | 32.4 + 2.1 |
Gallate-NPFF | 49 ± 4.2 |
NPFF | 22.5 ± 3.6 |